SCHEMBL7688050

SCHEMBL7688050

O=C(c1ccc(Br)cc1)c1cc(F)c(O)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.46
MAPT P10636 4/20 0.44
MAPK1 P28482 2/20 0.44
NPC1 O15118 1/20 0.44
HTT P42858 1/20 0.44
DGAT1 O75907 1/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43
CASP1 P29466 1/20 0.43
CYP2C19 P33261 1/20 0.43
LMNA P02545 3/20 0.42
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3469362 0.79 CASP3 (0.54) AKR1C3MAPTMAPK1NPC1HTT
SCHEMBL3468505 0.79 HSD17B1 (0.58) MAPTMAPK1CYP1A2CYP2C9HPGD
SCHEMBL7679390 0.78 KMT2A (0.54) AKR1C3MAPTMAPK1NPC1HTT
SCHEMBL5307521 0.77 CES2 (0.55) AKR1C3MAPTMAPK1NPC1HTT
SCHEMBL3467995 0.76 DGAT1 (0.56) AKR1C3MAPTNPC1HTTDGAT1
SCHEMBL17358779 0.75 MAPT (0.67) AKR1C3MAPTMAPK1NPC1HTT
SCHEMBL4214280 0.74 DGAT1 (0.58) AKR1C3MAPTMAPK1NPC1HTT
SCHEMBL3467964 0.74 AKR1C3 (0.47) AKR1C3MAPTMAPK1NPC1HTT
SCHEMBL25341126 0.73 HSD17B14 (0.50) DGAT1CYP1A2CYP2C9HPGDALOX15
SCHEMBL18993048 0.73 CA12 (0.50) MAPTKDM4EHSD17B1HSD17B2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed
US-5856503-A ANTICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 1999-01-05 US disclosed
EP-0778271-A2 Aminoalkyl-substituted benzo-heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed