SCHEMBL7706826

SCHEMBL7706826

Brc1cc(OCc2ccccc2)nc(OCc2ccccc2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
NUDT1 P36639 1/20 0.46
MAOB P27338 1/20 0.44
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43
GABRA5 P31644 2/20 0.43
GABRA3 P34903 2/20 0.43
ALOX5 P09917 2/20 0.42
PTGES O14684 1/20 0.40
HRH4 Q9H3N8 1/20 0.40
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
GABRA4 P48169 1/20 0.39
GABRE P78334 1/20 0.39
GABRA6 Q16445 1/20 0.39
GABRG1 Q8N1C3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8668544 0.90 MAOB (0.49) ALDH1A1MAOBGABRG2GABRB3GABRA5
SCHEMBL4270551 0.88 NUDT1 (0.51) ALDH1A1NUDT1MAOBGABRG2GABRB3
SCHEMBL1564355 0.80 ALDH1A1 (0.64) ALDH1A1NUDT1HRH4HTTLMNA
SCHEMBL8384805 0.80 PIN1 (0.47) ALDH1A1NUDT1ALOX5PTGESHRH4
SCHEMBL8871300 0.79 ALDH1A1 (0.59) ALDH1A1NUDT1MAOBALOX5HTT
SCHEMBL8561075 0.78 ALOX5 (0.48) ALDH1A1NUDT1MAOBGABRG2GABRB3
SCHEMBL11009131 0.78 TSHR (0.52) MAOBALOX5HTTLMNACYP3A4
SCHEMBL8565553 0.77 MRGPRX4 (0.45) ALDH1A1MAOBL3MBTL1GAA
SCHEMBL8669447 0.77 L3MBTL1 (0.45) ALDH1A1MAOBL3MBTL1GAA
SCHEMBL17995530 0.76 NUDT1 (0.46) ALDH1A1NUDT1ALOX5PTGESHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37623-E1 PHENYLTHIO AND PHENYLSELENO PYRIMIDINE ANALOGS el Kouni, Mahmoud H. 2002-04-02 US disclosed
EP-0725641-B1 NOVEL INHIBITORS OF URIDINE PHOSPHORYLASE (UrdPase) AND DIHYDROURACIL DEHYDROGENASE (DHUDase) EL KOUNI MAHMOUD H (US) 2000-12-13 EP disclosed
US-5721241-A PYRIMIDINE COMPOUND USEFUL TO DISRUPT VIRAL, CANCER, FUNGAL, PARASITE OR BACTERIAL REPLICATION AND DIHYDROURACIL DEHYDROGENASE OR URIDINE PHOSPHORYLASE INHIBITORS el Kouni, Mahmoud H. (US) 1998-02-24 US disclosed
EP-0725641-A4 1996-09-04 EP disclosed
EP-0725641-A1 NOVEL ENZYME INHIBITORS, THEIR SYNTHESIS, AND METHODS FOR USE El Kouni, Mahmoud H. (US) 1996-08-14 EP disclosed
US-5476855-A Pyrimidine analogs and nucleosides el Kouni, Mahmoud H. (US) 1995-12-19 US disclosed
WO-1995012400-A1 NOVEL ENZYME INHIBITORS, THEIR SYNTHESIS, AND METHODS FOR USE UAB RESEARCH FOUNDATION (US) 1995-05-11 WO disclosed