SCHEMBL7715098

SCHEMBL7715098

CC(C)(C)[Si](Oc1ccc2c(c1)C(N)CC2)(c1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACHE P22303 11/20 0.48
KDM1A O60341 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7263724 1.00 ACHE (0.48) ACHEKDM1AMAOAMAOBCYP19A1
SCHEMBL7259713 0.85 HCRTR1 (0.39) ACHEKDM1AMAOAMAOBCYP19A1
SCHEMBL7715113 0.85 HCRTR1 (0.39) ACHEKDM1AMAOAMAOBCYP19A1
SCHEMBL7717533 0.81 MTNR1B (0.35) ACHE
SCHEMBL7717534 0.81 MTNR1B (0.35) ACHE
SCHEMBL8620705 0.81 MTNR1A (0.34) ACHEKDM1AMAOAMAOB
SCHEMBL8617783 0.78 MTNR1A (0.39) ACHEKDM1AMAOAMAOB
SCHEMBL8636781 0.77 MAPK1 (0.36) ACHEKDM1AMAOAMAOB
SCHEMBL178121 0.76 PPARA (0.38) CYP19A1
SCHEMBL8647745 0.74 MAPK1 (0.39) ACHEKDM1AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441017-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2002-08-27 US disclosed
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed