SCHEMBL7732470

SCHEMBL7732470

N#Cc1ccc(C(=O)CCC2CCN(OC(=O)C(F)(F)F)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.48
BCHE P06276 2/20 0.42
ACHE P22303 2/20 0.42
HTR1A P08908 6/20 0.41
SLC6A4 P31645 5/20 0.40
GSK3B P49841 1/20 0.40
CHRM4 P08173 1/20 0.39
DRD2 P14416 1/20 0.39
HTR2A P28223 1/20 0.39
HTR7 P34969 1/20 0.39
HRH1 P35367 1/20 0.39
DRD3 P35462 1/20 0.39
HTR2B P41595 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7734278 0.85 DRD2 (0.46) SIGMAR1BCHEACHEHTR1ADRD2
SCHEMBL7723274 0.84 ACHE (0.59) SIGMAR1BCHEACHE
SCHEMBL17064427 0.81 SIGMAR1 (0.56) SIGMAR1BCHEACHEHTR1ASLC6A4
SCHEMBL7736003 0.79 MEN1 (0.48) SIGMAR1HTR1ADRD2HTR2ADRD3
SCHEMBL7723348 0.78 GPR119 (0.60) SIGMAR1
Trifluoroacetic Acid SCHEMBL7732466 0.77 KMT2A (0.45) SIGMAR1BCHEACHEHTR1ASLC6A4
SCHEMBL6475939 0.73 HSD11B1 (0.35)
SCHEMBL14790689 0.73 USP30 (0.39) CHRM4
SCHEMBL6475659 0.71 HSD11B1 (0.34)
SCHEMBL7731608 0.71 HDAC2 (0.40) HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399619-B1 PREVENTION AND TREATMENT OF AIDS AND VIRAL INFECTION BY HIV MERCK & CO., INC. 2002-06-04 US disclosed