SCHEMBL7737686

SCHEMBL7737686

COC(=O)CCc1cccc2c1OCC(=O)N2CCSC(C)(c1ccccc1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
TSHR P16473 3/20 0.38
HSD17B10 Q99714 2/20 0.38
MAPT P10636 1/20 0.38
HTR1A P08908 3/20 0.37
HTR1D P28221 3/20 0.37
HTR1B P28222 3/20 0.37
SLC6A4 P31645 3/20 0.37
KCNH2 Q12809 3/20 0.37
POLB P06746 1/20 0.37
CBX7 O95931 1/20 0.36
CDYL2 Q8N8U2 1/20 0.36
CDYL Q9Y232 1/20 0.36
CDY1; CDY1B Q9Y6F8 1/20 0.36
NMT1 P30419 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TP53 P04637 1/20 0.36
CHRM1 P11229 3/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7739735 0.91 HTR1A (0.39) ALDH1A1HTR1AHTR1DHTR1BSLC6A4
SCHEMBL7736480 0.82 ALDH1A1 (0.41) ALDH1A1TSHRHSD17B10MAPTHTR1A
SCHEMBL7737346 0.79 PTGIR (0.49) ALDH1A1TSHRHSD17B10POLBMEN1
SCHEMBL27688254 0.71 KMT2A (0.44) ALDH1A1TSHRHTR1AHTR1DHTR1B
SCHEMBL4969042 0.69 HSD17B10 (0.46) ALDH1A1TSHRHSD17B10MAPTPOLB
SCHEMBL27707632 0.67 KMT2A (0.44) ALDH1A1TSHRPOLBCBX7CDYL2
SCHEMBL7737376 0.66 TBXA2R (0.48) ALDH1A1POLBTBXA2RPTGIR
SCHEMBL7737236 0.65 TBXA2R (0.48) ALDH1A1POLBTBXA2RPTGIR
SCHEMBL7739672 0.64 KDM4E (0.38) ALDH1A1MAPTPOLBMEN1KMT2A
SCHEMBL7737187 0.64 HTR6 (0.41) ALDH1A1MAPTHTR1AKCNH2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407096-B1 1,4-BENZOTHIAZINE AND 1,4-BENZOXAZINE DERIVATIVES; HYPOTENSIVE, ANTIISCHEMIC, ANTIALLERGEN, ANTIASTHMATIC AND ANTICOAGULANT AGENTS; CARDIOVASCULAR DISORDERS TORAY INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1028113-A1 FUSED BENZENE HETEROCYCLE DERIVATIVES AND UTILIZATION THEREOF TORAY INDUSTRIES, INC. (JP) 2000-08-16 EP disclosed