SCHEMBL7739634

SCHEMBL7739634

CC(C)(C)OC(=O)C(N)(C(=O)OC(C)(C)C)c1cc(NC(N)=S)ccc1-n1cccc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
GAA P10253 3/20 0.36
KMT2A Q03164 2/20 0.35
CYP1A2 P05177 1/20 0.35
NR1I3 Q14994 1/20 0.34
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32
KCNH2 Q12809 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
ALOX12 P18054 1/20 0.31
CYP2C19 P33261 1/20 0.31
NPC1 O15118 2/20 0.31
MAPT P10636 2/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
PARP14 Q460N5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7734178 0.79 NTRK1 (0.35) ALDH1A1GAAKMT2ACYP1A2KDM4E
SCHEMBL7739635 0.76 ALDH1A1 (0.37) ALDH1A1GAAKMT2ACYP1A2NR1I3
SCHEMBL12071196 0.66 CYP17A1 (0.51) ALDH1A1GAAKMT2ACYP3A4CYP2D6
SCHEMBL27494826 0.66 ALDH1A1 (0.41) ALDH1A1GAAKMT2ACYP3A4CYP2D6
SCHEMBL6676211 0.65 ALDH1A1 (0.58) ALDH1A1GAAKMT2ACYP1A2KDM4E
SCHEMBL7740420 0.65 SYK (0.37) ALDH1A1GAAKMT2AKDM4EKCNH2
SCHEMBL7740422 0.64 SYK (0.40) ALDH1A1GAAKMT2AMAPTRAB9A
SCHEMBL27477483 0.64 KIF11 (0.42) ALDH1A1GAAKMT2ACYP3A4CYP2D6
SCHEMBL6675178 0.63 KDM4E (0.44) ALDH1A1GAAKMT2ANR1I3KDM4E
SCHEMBL6675941 0.62 KDM4E (0.43) ALDH1A1GAAKMT2ACYP1A2NR1I3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed