SCHEMBL7740476

SCHEMBL7740476

CCSC(N)=Nc1ccc(-n2cc(C)cn2)c(CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 18/20 0.38
NOS3 P29474 16/20 0.38
NOS2 P35228 16/20 0.38
HDAC10 Q969S8 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7740427 0.85 NOS1 (0.38) NOS1NOS3NOS2
SCHEMBL7740469 0.80 HDAC6 (0.34) HDAC10HDAC6CA12CA1CA2
SCHEMBL7738859 0.75 HDAC6 (0.36) HDAC10HDAC6CA12CA1CA2
SCHEMBL7734201 0.69 SYK (0.33) NOS1NOS3NOS2CA12CA1
SCHEMBL7742144 0.66 NOS1 (0.42) NOS1NOS3NOS2
SCHEMBL7734258 0.66 TDO2 (0.35)
SCHEMBL7740426 0.66 PDK1 (0.40) HDAC10HDAC6CA12CA1CA2
SCHEMBL7740424 0.65 MEN1 (0.36) HDAC10HDAC6
SCHEMBL29971591 0.64 CA12 (0.38) HDAC10HDAC6CA12CA1CA2
SCHEMBL18805717 0.64 CA12 (0.38) HDAC10HDAC6CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed