SCHEMBL7738859

SCHEMBL7738859

Cc1cnn(-c2ccc(NC#N)cc2CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.36
HDAC10 Q969S8 1/20 0.36
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
HDAC1 Q13547 1/20 0.35
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
CA12 O43570 1/20 0.34
AR P10275 2/20 0.34
NAMPT P43490 2/20 0.34
PRMT5 O14744 3/20 0.34
WDR77 Q9BQA1 3/20 0.34
NSD2 O96028 1/20 0.34
PIK3CA P42336 1/20 0.33
PIK3CG P48736 1/20 0.33
SCD O00767 1/20 0.33
SETDB1 Q15047 1/20 0.33
RAF1 P04049 1/20 0.33
BRAF P15056 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7740478 0.83 SYK (0.37) HDAC6HDAC10JAK2JAK1HDAC1
SCHEMBL7740469 0.81 HDAC6 (0.34) HDAC6HDAC10HDAC1CA1CA2
SCHEMBL7740476 0.75 NOS1 (0.38) HDAC6HDAC10CA1CA2CA9
SCHEMBL7740422 0.67 SYK (0.40) HDAC6HDAC10NAMPTBRD4MAPKAPK2
SCHEMBL26696901 0.67 RXFP1 (0.43) HDAC6HDAC10CA1CA2CA9
SCHEMBL7740426 0.65 PDK1 (0.40) HDAC6HDAC10CA1CA2CA9
SCHEMBL7734258 0.65 TDO2 (0.35) PIK3CAPIK3CG
SCHEMBL7738995 0.65 JAK2 (0.35) JAK2JAK1CA1CA2CA9
SCHEMBL7740424 0.65 MEN1 (0.36) HDAC6HDAC10NAMPTBRD4
SCHEMBL30419282 0.64 ATR (0.55) NAMPTSCDMAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed