SCHEMBL7747435

SCHEMBL7747435

O=C1Nc2ccc(Cl)cc2C2(CCN(C3CCN(C(=O)N4C(=O)OC[C@@H]4c4ccc(F)c(F)c4)CC3)CC2)O1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 2/20 0.39
ADRA1A P35348 2/20 0.39
ADRA1B P35368 2/20 0.39
AVPR1A P37288 1/20 0.37
PSEN1 P49768 2/20 0.36
PSEN2 P49810 2/20 0.36
APH1B Q8WW43 2/20 0.36
NCSTN Q92542 2/20 0.36
APH1A Q96BI3 2/20 0.36
PSENEN Q9NZ42 2/20 0.36
F11 P03951 11/20 0.36
CALCRL Q16602 2/20 0.36
ELOVL6 Q9H5J4 1/20 0.35
KLKB1 P03952 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7747425 0.79 ADRA1A (0.49) ADRA1DADRA1AADRA1B
SCHEMBL7743435 0.75 CCR2 (0.39) ADRA1DADRA1AADRA1BAVPR1AF11
SCHEMBL7743434 0.75 CCR2 (0.39) ADRA1DADRA1AADRA1BAVPR1AF11
SCHEMBL7747406 0.73 HRH3 (0.44) AVPR1AF11CALCRLELOVL6
SCHEMBL6965725 0.69 ADRA1D (0.44) ADRA1DADRA1AADRA1B
SCHEMBL7748936 0.68 CCR2 (0.43) ADRA1DADRA1AADRA1B
SCHEMBL3275750 0.65 CALCRL (0.51) AVPR1ACALCRL
SCHEMBL10952538 0.65 AVPR1A (0.47) AVPR1AF11
SCHEMBL5660885 0.65 MTOR (0.37) ADRA1DADRA1AADRA1B
SCHEMBL6082708 0.65 MTOR (0.37) ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001022919-A2 SPIRO[BICYCLIC -AZACYCLOALKYL AND -CYCLOALKYL] DERIVATIVES AND USES THEREOF MERCK & CO., INC. (US) 2001-04-05 WO disclosed