SCHEMBL7781180

SCHEMBL7781180

N=C(N)NN(c1cccc(C(CC(=O)O)NC(=O)c2ccc(C(F)(F)F)cc2)c1)S(=O)(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EEF2K O00418 3/20 0.46
CTSA P10619 5/20 0.44
KCNQ3 O43525 2/20 0.42
KCNQ2 O43526 2/20 0.42
ITGB3 P05106 4/20 0.40
ITGA2B P08514 4/20 0.40
WDR5 P61964 1/20 0.39
KCNA5 P22460 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
F10 P00742 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7194899 0.92 ITGB3 (0.44) CTSAITGB3ITGA2BF10
SCHEMBL7790178 0.91 CTSA (0.41) EEF2KCTSAITGB3ITGA2BF10
SCHEMBL7781206 0.90 ITGB3 (0.42) CTSAITGB3ITGA2BF10
SCHEMBL7788355 0.90 MMP12 (0.47) KCNQ3KCNQ2ITGB3ITGA2BWDR5
SCHEMBL7789969 0.90 CYP26A1 (0.42) CTSAITGB3ITGA2BF10
SCHEMBL7785658 0.87 LMNA (0.44) CTSAITGB3ITGA2BF10
SCHEMBL7788749 0.87 ITGB3 (0.44) CTSAITGB3ITGA2B
SCHEMBL7786214 0.86 S1PR3 (0.41) CTSAITGB3ITGA2B
SCHEMBL7786241 0.85 CTSA (0.46) CTSAITGB3ITGA2B
SCHEMBL7790073 0.85 CYP26A1 (0.46) CTSAITGB3ITGA2BF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147079-A2 BETA-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS Bayer Aktiengesellschaft (DE) 2001-10-24 EP disclosed
WO-2000041469-A2 β-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2000-07-20 WO disclosed