SCHEMBL7781206

SCHEMBL7781206

N=C(N)NN(c1cccc(C(CC(=O)O)NC(=O)c2ccc(-c3ccccc3)cc2)c1)S(=O)(=O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.42
ITGA2B P08514 2/20 0.42
F10 P00742 1/20 0.42
SUCNR1 Q9BXA5 2/20 0.41
MMP12 P39900 2/20 0.41
MMP3 P08254 1/20 0.40
MMP9 P14780 1/20 0.40
MMP8 P22894 1/20 0.40
MMP13 P45452 1/20 0.40
RPS6KA5 O75582 2/20 0.39
AKT1 P31749 2/20 0.39
GSK3B P49841 2/20 0.39
NEK4 P51957 2/20 0.39
PRKCD Q05655 2/20 0.39
PRKG2 Q13237 2/20 0.39
ROCK1 Q13464 2/20 0.39
PRKG1 Q13976 2/20 0.39
PKN2 Q16513 2/20 0.39
CLK4 Q9HAZ1 2/20 0.39
UTS2R Q9UKP6 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7194899 0.94 ITGB3 (0.44) ITGB3ITGA2BF10MAPK1CTSA
SCHEMBL7789969 0.92 CYP26A1 (0.42) ITGB3ITGA2BF10ROCK1UTS2R
SCHEMBL7790178 0.92 CTSA (0.41) ITGB3ITGA2BF10MMP12MAPK1
SCHEMBL7781180 0.90 EEF2K (0.46) ITGB3ITGA2BF10CTSA
SCHEMBL7785658 0.90 LMNA (0.44) ITGB3ITGA2BF10RPS6KA5AKT1
SCHEMBL7788749 0.89 ITGB3 (0.44) ITGB3ITGA2BUTS2RCTSAMEN1
SCHEMBL7786214 0.89 S1PR3 (0.41) ITGB3ITGA2BCTSACA1MEN1
SCHEMBL7786241 0.88 CTSA (0.46) ITGB3ITGA2BSUCNR1CTSAMEN1
SCHEMBL7790073 0.88 CYP26A1 (0.46) ITGB3ITGA2BF10ROCK1ROCK2
SCHEMBL7788355 0.87 MMP12 (0.47) ITGB3ITGA2BF10MMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147079-A2 BETA-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS Bayer Aktiengesellschaft (DE) 2001-10-24 EP disclosed
WO-2000041469-A2 β-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2000-07-20 WO disclosed