SCHEMBL7786214

SCHEMBL7786214

N=C(N)NN(c1cccc(C(CC(=O)O)NC(=O)c2ccc(Cl)c(Cl)c2)c1)S(=O)(=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 5/20 0.41
CTSA P10619 5/20 0.41
CYP26A1 O43174 3/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
S1PR4 O95977 3/20 0.40
S1PR2 O95136 2/20 0.40
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
GPR139 Q6DWJ6 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7786241 0.90 CTSA (0.46) S1PR3CTSAITGB3ITGA2BS1PR4
SCHEMBL7194899 0.90 ITGB3 (0.44) CTSACYP26A1ITGB3ITGA2BMEN1
SCHEMBL7788749 0.89 ITGB3 (0.44) CTSAITGB3ITGA2BCA2MEN1
SCHEMBL7781206 0.89 ITGB3 (0.42) CTSAITGB3ITGA2BCA1MEN1
SCHEMBL7789969 0.88 CYP26A1 (0.42) CTSACYP26A1ITGB3ITGA2BALDH1A1
SCHEMBL7790178 0.88 CTSA (0.41) CTSACYP26A1ITGB3ITGA2BMEN1
SCHEMBL7790073 0.87 CYP26A1 (0.46) CTSACYP26A1ITGB3ITGA2BGPR139
SCHEMBL7781180 0.86 EEF2K (0.46) CTSAITGB3ITGA2B
SCHEMBL7785658 0.85 LMNA (0.44) S1PR3CTSAITGB3ITGA2BCA2
SCHEMBL7785607 0.85 LMNA (0.46) S1PR3ITGB3GPR139MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147079-A2 BETA-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS Bayer Aktiengesellschaft (DE) 2001-10-24 EP disclosed
WO-2000041469-A2 β-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2000-07-20 WO disclosed