SCHEMBL7787602

SCHEMBL7787602

COc1ccc(C(NCCc2cccc(F)c2)c2cccc(N)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
LMNA P02545 2/20 0.44
GAA P10253 1/20 0.44
TAAR1 Q96RJ0 1/20 0.43
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
KMT2A Q03164 3/20 0.40
MAOB P27338 3/20 0.40
NOS1 P29475 2/20 0.39
MEN1 O00255 1/20 0.39
NOS3 P29474 1/20 0.39
MITF O75030 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789351 0.92 TDP1 (0.41) ALDH1A1LMNAGAACYP1A2CYP2D6
SCHEMBL7780362 0.89 TDP1 (0.50) ALDH1A1LMNAGAATDP1KMT2A
SCHEMBL7785046 0.89 TDP1 (0.49) ALDH1A1GAATAAR1TDP1KMT2A
SCHEMBL7789039 0.82 KMT2A (0.46) ALDH1A1LMNAGAAL3MBTL1TDP1
SCHEMBL7789152 0.82 SIGMAR1 (0.53) ALDH1A1LMNAGAATDP1KMT2A
SCHEMBL7787489 0.82 ALDH1A1 (0.39) ALDH1A1LMNAGAATAAR1CYP1A2
SCHEMBL7780337 0.78 ALDH1A1 (0.40) ALDH1A1LMNAGAATAAR1CYP1A2
SCHEMBL7780342 0.78 KMT2A (0.54) ALDH1A1LMNATDP1KMT2AMEN1
SCHEMBL7785107 0.77 ALDH1A1 (0.50) ALDH1A1LMNAGAACYP1A2CYP2D6
SCHEMBL7780790 0.77 ALDH1A1 (0.50) ALDH1A1LMNAGAACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329405-B1 AS ILEAL BILE ACID TRANSPORTER INHIBITOR, FOR THERAPY OF HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 2001-12-11 US disclosed
CN-1287117-A Cyclobutene derivatives, preparation method and therapeutic use thereof SANKYO CO (JP) 2001-03-14 CN disclosed
EP-1070703-A1 Cyclobutene derivatives Sankyo Company Limited (JP) 2001-01-24 EP disclosed