SCHEMBL7789876

SCHEMBL7789876

CCC(CO)NC(=O)c1cccc(-c2ccc3ccccc3c2C(N)=O)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 6/20 0.46
DYRK2 Q92630 6/20 0.46
DYRK1B Q9Y463 6/20 0.46
DYRK3 O43781 5/20 0.46
CCNA2 P20248 1/20 0.44
CDK2 P24941 1/20 0.44
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
HPGD P15428 1/20 0.42
F3 P13726 1/20 0.41
PPARG P37231 3/20 0.39
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7782141 0.88 HPGDS (0.47) DYRK1ADYRK1B
SCHEMBL7789847 0.85 PPARG (0.39) PPARG
SCHEMBL7782223 0.82 MEN1 (0.47) HPGDF3TAS1R3TAS1R1
SCHEMBL7782229 0.77 CAPN1 (0.51)
SCHEMBL7325294 0.76 KMO (0.49) HPGD
SCHEMBL7787012 0.75 ROCK2 (0.47) DYRK1ADYRK1BF3
SCHEMBL7790079 0.74 ROCK2 (0.43) DYRK1ADYRK1B
SCHEMBL722165 0.73 BCAT2 (0.47) HPGD
SCHEMBL7314496 0.71 PIN1 (0.48)
SCHEMBL7787042 0.71 DYRK1A (0.47) DYRK1ADYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed