SCHEMBL7797241

SCHEMBL7797241

COc1ccccc1-n1cc(-c2ccccc2)oc1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 3/20 0.46
HSD17B10 Q99714 3/20 0.46
CYP3A4 P08684 2/20 0.46
HPGD P15428 2/20 0.46
TP53 P04637 1/20 0.46
AR P10275 1/20 0.46
GAA P10253 2/20 0.44
MGLL Q99685 1/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ABCG2 Q9UNQ0 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ADORA3 P0DMS8 2/20 0.41
ADORA1 P30542 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6757704 0.80 MGLL (0.47) ALDH1A1KDM4EMAPTHSD17B10HPGD
SCHEMBL7944253 0.79 HTR7 (0.49) ALDH1A1KDM4E
SCHEMBL7807349 0.77 KDM4E (0.44) ALDH1A1KDM4EMAPTHSD17B10CYP3A4
SCHEMBL11668799 0.74 ASAH1 (0.42) ALDH1A1KDM4EMAPTHSD17B10CYP3A4
SCHEMBL7805538 0.73 ALDH1A1 (0.49) ALDH1A1KDM4EMAPTHSD17B10CYP3A4
SCHEMBL10059782 0.73 ALDH1A1 (0.49) ALDH1A1MAPTGAAMGLLNPC1
SCHEMBL7807340 0.70 ADORA3 (0.48) ALDH1A1KDM4EMAPTHSD17B10HPGD
SCHEMBL7981999 0.66 GAA (0.58) ALDH1A1KDM4EMAPTHPGDGAA
SCHEMBL3304455 0.66 ALDH1A1 (0.54) ALDH1A1KDM4EMAPTHSD17B10HPGD
SCHEMBL6560725 0.65 TUBB4A (0.46) ALDH1A1TP53GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6255327-B1 ANTIHYPOXC, ANTIISCHEMIC AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-03 US disclosed
EP-1071670-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-01-31 EP disclosed
WO-1999054314-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-28 WO disclosed