SCHEMBL7806505

SCHEMBL7806505

CCCCc1ccc2c(nc(OC)n2C)c1-c1cc(Cl)c(Cl)cc1Cl

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 3/20 0.32
HSD11B1 P28845 1/20 0.32
ELANE P08246 2/20 0.31
CTSG P08311 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
ERBB2 P04626 1/20 0.30
NPBWR1 P48145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817046 0.81 POLB (0.33) KDM4E
SCHEMBL7816658 0.76 CRHR1 (0.32) CRHR1
SCHEMBL7814352 0.66 HCAR1 (0.34)
SCHEMBL7813650 0.66 CYP11B2 (0.31)
SCHEMBL30098086 0.60 CNR2 (0.35) ELANECTSG
SCHEMBL21815186 0.58 SMN1; SMN2 (0.51)
SCHEMBL20467095 0.57 ALOX5 (0.41) ELANE
SCHEMBL19003636 0.56 ERBB2 (0.44) ERBB2
SCHEMBL20014473 0.56 OXER1 (0.47)
SCHEMBL21230758 0.56 ALOX5 (0.40) ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091941-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2001-04-18 EP claimed
WO-2000001675-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 2000-01-13 WO claimed