Water

Water

SCHEMBL78121

N=C1C=CC(=O)C=C1.O

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL59611 0.96
Sulfurous Acid SCHEMBL11527320 0.82 ALDH1A1 (0.44)
Benzoquinone SCHEMBL10610820 0.80 ALDH1A1 (0.89)
Benzoquinone SCHEMBL3656695 0.80 ALDH1A1 (0.89)
Naphthalene SCHEMBL6910660 0.80 MAOA (0.42)
Benzoquinone SCHEMBL28240806 0.76
SCHEMBL148004 0.76
Benzoquinone SCHEMBL18103 0.76
Benzoquinone SCHEMBL30679171 0.76
Benzoquinone SCHEMBL10506648 0.76 ALDH1A1 (1.00)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326943-B1 C-NITROSOANILINE COMPOUNDS AND THEIR BLENDS AS POLYMERIZATION INHIBITORS UNIROYAL CHEM CO INC (US) 2006-01-25 EP claimed
US-20040104146-A1 C-nitrosoaniline compounds and their blends as polymerization inhibitors UNIROYAL CHEMICAL COMPANY, INC. 2004-06-03 US claimed
US-20040106753-A1 C-nitrosoaniline compounds and their blends as polymerization inhibitors UNIROYAL CHEMICAL COMPANY, INC. 2004-06-03 US claimed
US-20040089586-A1 C-nitrosoaniline compounds and their blends as polymerization inhibitors UNIROYAL CHEMICAL COMPANY, INC. 2004-05-13 US claimed
EP-1326943-A2 C-NITROSOANILINE COMPOUNDS AND THEIR BLENDS AS POLYMERIZATION INHIBITORS Uniroyal Chemical Company, Inc. (US) 2003-07-16 EP claimed
US-20030047439-A1 C-nitrosoaniline compounds and their blends as polymerization inhibitors ADDIVANT USA, LLC 2003-03-13 US claimed
WO-2002033025-A2 C-NITROSOANILINE COMPOUNDS AND THEIR BLENDS AS POLYMERIZATION INHIBITORS UNIROYAL CHEMICAL COMPANY, INC. (US) 2002-04-25 WO claimed
US-8809431-B2 Process for stabilizing olefinically unsaturated monomers EVONIK DEGUSSA GMBH (DE) 2014-08-19 US disclosed
US-20120101295-A1 PROCESS FOR STABILIZING OLEFINICALLY UNSATURATED MONOMERS EVONIK DEGUSSA GMBH (DE) 2012-04-26 US disclosed
US-8128804-B2 Process for stabilizing olefinically unsaturated monomers EVONIK DEGUSSA GMBH (DE) 2012-03-06 US disclosed
US-20090114878-A1 PROCESS FOR STABILIZING OLEFINICALLY UNSATURATED MONOMERS EVONIK DEGUSSA GMBH (DE) 2009-05-07 US disclosed
US-7022220-B2 C-nitrosoaniline compounds and their blends as polymerization inhibitors UNIROYAL CHEMICAL COMPANY, INC. (US) 2006-04-04 US disclosed
EP-1326943-B1 C-NITROSOANILINE COMPOUNDS AND THEIR BLENDS AS POLYMERIZATION INHIBITORS UNIROYAL CHEM CO INC (US) 2006-01-25 EP disclosed
US-20040104146-A1 C-nitrosoaniline compounds and their blends as polymerization inhibitors UNIROYAL CHEMICAL COMPANY, INC. 2004-06-03 US disclosed
US-20040106753-A1 C-nitrosoaniline compounds and their blends as polymerization inhibitors UNIROYAL CHEMICAL COMPANY, INC. 2004-06-03 US disclosed
US-20040089586-A1 C-nitrosoaniline compounds and their blends as polymerization inhibitors UNIROYAL CHEMICAL COMPANY, INC. 2004-05-13 US disclosed
US-6685823-B2 INHIBITING THE PREMATURE POLYMERIZATION OF ETHYLENICALLY UNSATURATED MONOMERS BY ADDING COMPOUNDS SELECTED FROM C-NITROSOANILINE AND QUINONE IMINE OXIME COMPOUNDS UNIROYAL CHEMICAL COMPANY, INC. 2004-02-03 US disclosed
EP-1326943-A2 C-NITROSOANILINE COMPOUNDS AND THEIR BLENDS AS POLYMERIZATION INHIBITORS Uniroyal Chemical Company, Inc. (US) 2003-07-16 EP disclosed
US-20030047439-A1 C-nitrosoaniline compounds and their blends as polymerization inhibitors ADDIVANT USA, LLC 2003-03-13 US disclosed
WO-2002033025-A2 C-NITROSOANILINE COMPOUNDS AND THEIR BLENDS AS POLYMERIZATION INHIBITORS UNIROYAL CHEMICAL COMPANY, INC. (US) 2002-04-25 WO disclosed