SCHEMBL7816809

SCHEMBL7816809

O=C(O)c1cncc(O)c1C(=O)c1cc(Cl)ccc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
XDH P47989 3/20 0.40
SLC22A12 Q96S37 3/20 0.40
GRM5 P41594 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TGFBR1 P36897 1/20 0.39
GAA P10253 1/20 0.38
PKM P14618 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
ANO1 Q5XXA6 1/20 0.38
KMO O15229 2/20 0.37
KCNMA1 Q12791 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
TAS1R2 Q8TE23 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817359 0.84 KDM4E (0.45) ALDH1A1GRM5TGFBR1GAAMRGPRX4
SCHEMBL7812042 0.77 TGFBR1 (0.47) CA1CA2ALDH1A1TP53TSHR
SCHEMBL7804698 0.77 TGFBR1 (0.47) CA1CA2ALDH1A1TP53TSHR
SCHEMBL30396748 0.75 ALDH1A1 (0.65) CA1CA2ALDH1A1TP53TSHR
SCHEMBL283203 0.75 ALDH1A1 (0.65) CA1CA2ALDH1A1TP53TSHR
SCHEMBL7816890 0.73 CA1 (0.43) CA1CA2ALDH1A1TP53XDH
SCHEMBL28072667 0.73 ALDH1A1 (0.50) CA1CA2ALDH1A1TP53TSHR
SCHEMBL15241144 0.71 KMO (0.48) CA1CA2ALDH1A1TP53GRM5
SCHEMBL9435361 0.71 TGFBR1 (0.48) ALDH1A1TGFBR1
SCHEMBL28297856 0.71 KDM4E (0.41) CA1CA2ALDH1A1XDHSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750619-B1 HETERO-ANNULATED INDAZOLES NOVUSPHARMA SPA (IT) 2001-05-30 EP disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
EP-0750619-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA S.p.A. (IT) 1997-01-02 EP disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed