SCHEMBL7824904

SCHEMBL7824904

O=Cc1c(CCCI)[nH]c2cccc(Cl)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
GPR17 Q13304 1/20 0.36
ERCC5 P28715 1/20 0.35
FEN1 P39748 1/20 0.35
GRIN2D O15399 2/20 0.33
GRIN3B O60391 2/20 0.33
GRIN1 Q05586 2/20 0.33
GRIN2A Q12879 2/20 0.33
GRIN2B Q13224 2/20 0.33
GRIN2C Q14957 2/20 0.33
GRIN3A Q8TCU5 2/20 0.33
DYRK1A Q13627 1/20 0.33
GPR84 Q9NQS5 1/20 0.33
MCL1 Q07820 3/20 0.32
MET P08581 2/20 0.32
CHEK1 O14757 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834282 0.87 AHR (0.41) AHRMEN1ALDH1A1KMT2ATDP1
SCHEMBL29954948 0.74 MEN1 (0.52) AHRMEN1ALDH1A1KMT2ATDP1
SCHEMBL7493525 0.71 ALDH1A1 (0.48) AHRMEN1ALDH1A1KMT2ATDP1
SCHEMBL27784055 0.68 GPR17 (0.56) MEN1ALDH1A1KMT2ATDP1GPR17
SCHEMBL7835174 0.67 MAPT (0.42) MEN1ALDH1A1KMT2A
SCHEMBL7824030 0.67 SIRT1 (0.40) AHRALDH1A1KMT2ADYRK1AMET
SCHEMBL7834087 0.66 MPO (0.33) AHR
SCHEMBL28135012 0.65 GPR84 (0.36) AHRALDH1A1GPR84MCL1
SCHEMBL7836059 0.65 AHR (0.54) AHRMEN1ALDH1A1KMT2A
SCHEMBL28303266 0.65 MEN1 (0.41) AHRMEN1ALDH1A1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109813-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2001-06-27 EP disclosed
WO-2000012510-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2000-03-09 WO disclosed