SCHEMBL7828647

SCHEMBL7828647

CC(=O)N(CCCCN1CCN(c2cc3ccc(F)cc3s2)CC1)C(=O)C(C)C

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.38
DRD2 P14416 5/20 0.38
HTR2A P28223 3/20 0.38
FPR3 P25089 1/20 0.35
FPR2 P25090 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HTR7 P34969 2/20 0.35
KCNH2 Q12809 1/20 0.35
DRD3 P35462 2/20 0.35
DRD4 P21917 2/20 0.35
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7828641 0.81 HTR2A (0.54) HTR1ADRD2HTR2AHTR7DRD3
SCHEMBL31240335 0.61 DRD2 (0.45) HTR1ADRD2HTR2AHTR7KCNH2
SCHEMBL7830765 0.60 ADRA1A (0.67) HTR1ADRD2HTR2ADRD3DRD4
SCHEMBL9360288 0.60 ACHE (0.53) HTR1ADRD2HTR2AHTR7DRD3
SCHEMBL7824411 0.58 ADRA1A (0.70) HTR1ADRD2HTR2ADRD3DRD4
SCHEMBL10527898 0.58 HRH3 (0.52) HTR1ADRD2HTR2ADRD3DRD4
SCHEMBL4574733 0.58 DRD2 (0.57) HTR1ADRD2HTR2AKCNH2
SCHEMBL9428377 0.57 CCR5 (0.44) KCNH2
SCHEMBL13809609 0.55 HTR2A (0.40) HTR1ADRD2HTR2ARAB9ADRD4
SCHEMBL8011318 0.54 DRD2 (0.69) HTR1ADRD2HTR2AKCNH2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0732332-B1 Substituted benzothienylpiperazines, their use as medicaments, and processes for their preparation AVENTIS PHARMA INC (US) 2001-12-19 EP disclosed