SCHEMBL784140

SCHEMBL784140

NS(=O)(=O)c1cccnc1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 10/20 0.51
CA2 P00918 10/20 0.51
CA9 Q16790 8/20 0.51
MAPK1 P28482 1/20 0.51
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47
CA12 O43570 6/20 0.46
CA6 P23280 3/20 0.44
CA4 P22748 2/20 0.44
CA5A P35218 2/20 0.44
CA7 P43166 2/20 0.44
CA5B Q9Y2D0 2/20 0.44
CYP2C9 P11712 1/20 0.44
CA14 Q9ULX7 1/20 0.44
FTO Q9C0B1 1/20 0.44
LMNA P02545 2/20 0.43
TDP1 Q9NUW8 1/20 0.42
CTSL P07711 1/20 0.40
PTPRC P08575 1/20 0.40
CTSS P25774 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2565634 0.87 CA2 (0.50) CA1CA2CA9MAPK1CA12
Hydrochloric Acid SCHEMBL29970039 0.83 CA2 (0.53) CA1CA2CA9MAPK1PTGS2
SCHEMBL5850523 0.81 PTGS1 (0.47) PTGS1PTGS2LMNATDP1CTSL
SCHEMBL5700053 0.81 PTGS2 (0.59) PTGS1PTGS2LMNATDP1CTSL
SCHEMBL28216449 0.80 CA2 (0.47) CA1CA2CA9MAPK1PTGS1
SCHEMBL12474849 0.80 CA1 (0.47) CA1CA2CA9MAPK1PTGS1
SCHEMBL8514484 0.80 CA2 (0.50) CA1CA2CA9MAPK1CA12
SCHEMBL29233670 0.77 PTGS1 (0.44) CA1CA2CA9MAPK1PTGS1
SCHEMBL29718566 0.77 CA2 (0.47) CA1CA2CA9MAPK1CA12
SCHEMBL790692 0.76 CA1 (0.52) CA1CA2CA9MAPK1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108822002-A A kind of method of ultrasonic wave added synthesis N- aryl sulfonic acid amides 中南大学 2018-11-16 CN disclosed
CN-107922362-A 1,3, 4-oxadiazole sulfonamide derivative compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions containing the same 株式会社钟根堂 2018-04-17 CN disclosed
US-8841302-B2 HCV inhibitor and therapeutic agent combinations PTC THERAPEUTICS, INC. (US) 2014-09-23 US disclosed
US-8735414-B2 Indole derivatives and methods for antiviral treatment PTC THERAPEUTICS, INC. (US) 2014-05-27 US disclosed
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
US-20120184574-A1 INDOLE DERIVATIVES AND METHODS FOR ANTIVIRAL TREATMENT PTC THERAPEUTICS, INC. (US) 2012-07-19 US disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
US-20120070412-A1 HCV Inhibitor and Therapeutic Agent Combinations PTC THERAPEUTICS, INC. (US) 2012-03-22 US disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
CN-1097051-C N-heteroaryl-pyridinesulfonamide derivatives and their use as endothelin antagonists ZENECA LTD (GB) 2002-12-25 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120070412-A1 HCV Inhibitor and Therapeutic Agent Combinations HAVCR2, SERPINB1, ENPEP CA1 4155/4885CA2 3704/4885CA9 3940/4885
US-20120184574-A1 INDOLE DERIVATIVES AND METHODS FOR ANTIVIRAL TREATMENT IDO1, IRF3, MAVS CA1 4515/4885CA2 3559/4885CA9 4223/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.