SCHEMBL7844124

SCHEMBL7844124

O=C(c1ccno1)N1CCc2c([nH]c3ccc(Br)cc23)C1C1(C(=O)O)CCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.40
ABCG2 Q9UNQ0 4/20 0.38
DHODH Q02127 1/20 0.36
CYP2D6 P10635 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
BAZ2B Q9UIF8 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
PKM P14618 2/20 0.34
SIRT1 Q96EB6 1/20 0.34
ABCB1 P08183 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
TRPV1 Q8NER1 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7855705 0.90 SIRT1 (0.45) KIF11SIRT1ALDH1A1MAPT
SCHEMBL7683405 0.88 KIF11 (0.38) KIF11ABCG2KDM4ENPSR1ALDH1A1
SCHEMBL7851436 0.82 ABCG2 (0.42) KIF11ABCG2DHODHCYP2D6OPRM1
SCHEMBL7683829 0.79 LMNA (0.46) KIF11KDM4EHTR2AHTR2CSIRT1
SCHEMBL7843396 0.75 TP53 (0.57) KIF11ABCG2KDM4ESIRT1ABCB1
SCHEMBL7847564 0.75 SIRT1 (0.47) KIF11ABCG2DHODHHTR2AHTR2C
SCHEMBL7855327 0.75 KIF11 (0.47) KIF11ABCG2SIRT1ABCB1ALDH1A1
SCHEMBL7854615 0.74 KIF11 (0.52) KIF11ABCG2SIRT1ABCB1ALDH1A1
SCHEMBL7852593 0.74 LMNA (0.46) KIF11SIRT1MAPT
SCHEMBL7853673 0.73 MAPKAPK2 (0.49) ABCG2SIRT1ABCB1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070716-A1 Beta-carboline derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2001-01-24 EP disclosed