SCHEMBL7860396

SCHEMBL7860396

COC(=O)C(CCN1C(=O)c2ccccc2C1=O)(CC(=O)c1ccc(OC)cc1)C(=O)OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.60
GAA P10253 2/20 0.56
HSD17B10 Q99714 2/20 0.50
RAB9A P51151 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
ALDH1A1 P00352 3/20 0.48
POLB P06746 3/20 0.48
APEX1 P27695 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
MMP2 P08253 2/20 0.48
MMP9 P14780 2/20 0.48
RPS6KA2 Q15349 1/20 0.46
CASP3 P42574 1/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP2D6 P10635 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7574583 0.77 MEN1 (0.46) NPC1GAARAB9AMEN1KMT2A
SCHEMBL6296941 0.77 NPC1 (0.42) NPC1GAAHSD17B10RAB9AMEN1
SCHEMBL6293053 0.76 MMP2 (0.43) NPC1GAAALDH1A1MMP2MMP9
SCHEMBL1609155 0.76 NPC1 (1.00) NPC1GAAHSD17B10RAB9AMEN1
SCHEMBL14288291 0.76 NPC1 (0.69) NPC1GAAHSD17B10RAB9AMEN1
SCHEMBL8531541 0.75 POLB (0.56) HSD17B10RAB9AMEN1KMT2AALDH1A1
SCHEMBL17163193 0.75 SMN1; SMN2 (0.47) GAAHSD17B10MEN1KMT2AALDH1A1
SCHEMBL7862778 0.74 GSK3B (0.59) NPC1MEN1KMT2AALDH1A1POLB
SCHEMBL7861865 0.73 THRA (0.41) GAAHSD17B10RAB9APOLBAPEX1
SCHEMBL7861710 0.73 GSK3B (0.49) NPC1GAAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923529-B1 SUBSTITUTE 4-ARYLBUTYRIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS BAYER AG (US) 2001-09-19 EP disclosed
EP-0923529-A1 SUBSITUTE 4-ARYLBUTYRIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS Bayer Corporation (US) 1999-06-23 EP disclosed
US-5863915-A ENZYME INHIBITORS FOR BONES AND JOINTS BAYER CORPORATION (US) 1999-01-26 US disclosed
WO-1997043237-A1 SUBSITUTE 4-ARYLBUTYRIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS BAYER CORPORATION (US) 1997-11-20 WO disclosed