SCHEMBL789718

SCHEMBL789718

CSc1c(-c2ccccc2)c(N)nc2ccc(I)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 3/20 0.41
CYP1A2 P05177 3/20 0.41
CYP1B1 Q16678 2/20 0.41
DHFR P00374 3/20 0.39
HEXA P06865 1/20 0.39
HEXB P07686 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTPN1 P18031 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
DHODH Q02127 1/20 0.35
NR1I3 Q14994 1/20 0.35
APP P05067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789402 0.78 CYP1A2 (0.41) CYP1A1CYP1A2CYP1B1DHFRHEXA
SCHEMBL790933 0.78 APP (0.47) CYP1A1CYP1A2CYP1B1DHFRHEXA
SCHEMBL790753 0.76 CYP1A2 (0.37) CYP1A1CYP1A2CYP1B1DHFRHEXA
SCHEMBL790609 0.75 LMNA (0.48) DHODH
SCHEMBL790759 0.75 KDM4E (0.47) KDM4EALDH1A1
SCHEMBL27556561 0.73 CYP1A1 (0.69) CYP1A1CYP1A2CYP1B1MAPTALDH1A1
SCHEMBL29058866 0.69 ESR1 (0.64) CYP1A1CYP1A2CYP1B1KDM4EMAPT
SCHEMBL16645243 0.68 ESR1 (0.43) CYP1A2KDM4EMAPTALDH1A1GAA
SCHEMBL28041367 0.67 KDM4E (0.50) CYP1A1CYP1A2CYP1B1KDM4EMAPT
SCHEMBL12974183 0.66 DHODH (0.47) KDM4EMAPTTDP1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed