SCHEMBL790753

SCHEMBL790753

C[S+]([O-])c1c(-c2ccccc2)c(N)nc2ccc(I)cc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.37
CYP1A1 P04798 2/20 0.37
CYP1B1 Q16678 2/20 0.37
MAPK1 P28482 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DHFR P00374 3/20 0.35
HEXA P06865 1/20 0.35
HEXB P07686 1/20 0.35
ESR1 P03372 2/20 0.33
ESR2 Q92731 2/20 0.33
APP P05067 1/20 0.33
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789402 0.76 CYP1A2 (0.41) CYP1A2CYP1A1CYP1B1MAPK1KDM4E
SCHEMBL790933 0.76 APP (0.47) CYP1A2CYP1A1CYP1B1MAPK1KDM4E
SCHEMBL789718 0.76 CYP1A1 (0.41) CYP1A2CYP1A1CYP1B1MAPK1KDM4E
SCHEMBL790609 0.73 LMNA (0.48) PTGFR
SCHEMBL790759 0.73 KDM4E (0.47) KDM4ENPSR1
SCHEMBL29058866 0.70 ESR1 (0.64) CYP1A2CYP1A1CYP1B1KDM4EMAPT
SCHEMBL27556561 0.68 CYP1A1 (0.69) CYP1A2CYP1A1CYP1B1MAPT
SCHEMBL28041367 0.65 KDM4E (0.50) CYP1A2CYP1A1CYP1B1MAPK1KDM4E
SCHEMBL390680 0.64 ESR1 (0.41) CYP1A2CYP1A1CYP1B1MAPK1KDM4E
SCHEMBL28041598 0.63 KDM4E (0.56) CYP1A2MAPK1KDM4EMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed