SCHEMBL790093

SCHEMBL790093

COc1ccc(CNc2nc3ccc(-c4cccc(NC(=O)c5cccnc5)c4)cc3cc2-c2ccc(N3CCOCC3)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.48
TP53 P04637 2/20 0.48
PIK3CA P42336 1/20 0.46
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
MAPT P10636 4/20 0.45
LMNA P02545 2/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
KDR P35968 1/20 0.45
MAPK14 Q16539 2/20 0.44
USP2 O75604 1/20 0.44
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TSHR P16473 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789915 0.93 RAB9A (0.50) SMN1; SMN2TP53RAB9ANPC1MAPT
SCHEMBL790392 0.90 KDR (0.48) SMN1; SMN2TP53RAB9ANPC1MAPT
SCHEMBL791145 0.88 KDR (0.46) TP53PIK3CARAB9ANPC1MAPT
SCHEMBL790416 0.85 MRGPRX4 (0.50) PIK3CARAB9AMAPTLMNAMEN1
SCHEMBL790646 0.85 KDR (0.47) RAB9AMAPTLMNAMEN1KMT2A
SCHEMBL789511 0.81 SMN1; SMN2 (0.59) SMN1; SMN2TP53PIK3CARAB9ANPC1
SCHEMBL791199 0.81 RAB9A (0.50) PIK3CARAB9ALMNAKDRSTAT6
SCHEMBL790621 0.80 KDR (0.46) RAB9ANPC1MAPTLMNAMEN1
SCHEMBL789889 0.78 RAB9A (0.48) PIK3CARAB9AKDRMAPK1STAT6
SCHEMBL790788 0.72 NPC1 (0.54) RAB9ANPC1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed