SCHEMBL7905966

SCHEMBL7905966

COc1cccc(-c2nnc(-n3nc(N4CCCCC4)nc3N)s2)c1OCCCN1CCOCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.49
TSHR P16473 1/20 0.49
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
KMT2A Q03164 1/20 0.40
HRH3 Q9Y5N1 2/20 0.38
KCNH2 Q12809 1/20 0.38
ATM Q13315 1/20 0.38
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
POLB P06746 1/20 0.37
AXL P30530 1/20 0.37
BACE1 P56817 1/20 0.37
TLR9 Q9NR96 2/20 0.37
TLR7 Q9NYK1 2/20 0.37
QPCT Q16769 1/20 0.36
QPCTL Q9NXS2 1/20 0.36
FLT3 P36888 1/20 0.36
MGAM O43451 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7904632 0.87 HRH3 (0.41) CYP2D6TSHRALDH1A1MEN1CYP1A2
SCHEMBL7904007 0.87 USP2 (0.40) ALDH1A1MEN1KMT2AHRH3KDM4E
SCHEMBL7904674 0.84 QPCT (0.51) CYP2D6TSHRHRH3ATMKDM4E
SCHEMBL7905773 0.81 BACE1 (0.39) CYP2D6ALDH1A1CYP1A2HRH3KDM4E
SCHEMBL7896424 0.80 ALDH1A1 (0.42) ALDH1A1MEN1KMT2AHRH3KCNH2
SCHEMBL7908545 0.78 PRKDC (0.39) CYP2D6CYP1A2KDM4ETDP1POLB
SCHEMBL7896551 0.76 CNR2 (0.36) TSHRMEN1KMT2AHRH3KDM4E
SCHEMBL7905780 0.75 HRH3 (0.40) TSHRALDH1A1MEN1KMT2AHRH3
SCHEMBL7896411 0.75 USP2 (0.43) CYP2D6TSHRALDH1A1CYP1A2HRH3
SCHEMBL7908481 0.75 PIK3CB (0.44) TSHRMEN1KMT2AHRH3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191152-B1 CARDIOVASCULAR DISORDERS, NERVOUS SYSTEM DISORDERS EGIS GYÓGYSZERGYAR RT. (HU) 2001-02-20 US disclosed