SCHEMBL7921611

SCHEMBL7921611

COCC(=O)[C@](CC(C)C)(C(=O)NNCC(C)C)[C@H](CC=Cc1ccccc1)C(=O)NO

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.35
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
HTR2A P28223 3/20 0.32
USP2 O75604 1/20 0.32
TSHR P16473 1/20 0.32
CTSC P53634 1/20 0.32
GAA P10253 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GHSR Q92847 2/20 0.31
GRIK1 P39086 2/20 0.30
GRIK2 Q13002 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7931036 0.72 GHSR (0.32) GHSR
SCHEMBL6942735 0.67 ADAM17 (0.42) ADAM17MMP1MMP9MMP13HTR2A
SCHEMBL7957560 0.67 GHSR (0.37) ADAM17HTR2ATSHRCTSCGHSR
SCHEMBL6940930 0.66 ADAM17 (0.40) ADAM17MMP1MMP9MMP13CTSC
SCHEMBL7931077 0.65 ADAM17 (0.34) ADAM17HTR2ACTSCGAASMN1; SMN2
SCHEMBL6942460 0.64 ADAM17 (0.46) ADAM17MMP1HTR2ACTSCGRIK1
SCHEMBL6945084 0.64 ADAM17 (0.42) ADAM17MMP1MMP9MMP13HTR2A
SCHEMBL7103597 0.62 ADAM17 (0.48) ADAM17MMP1MMP9MMP13HTR2A
SCHEMBL7107632 0.62 ADAM17 (0.48) ADAM17MMP1MMP9MMP13HTR2A
SCHEMBL27947171 0.61 HTR2A (0.53) HTR2ACTSCGRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed