SCHEMBL7922258

SCHEMBL7922258

NC=S.O=C(Cn1nnc(-c2cc(Cl)cc(Cl)c2)n1)NNc1ccc(Cl)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.48
ALDH1A1 P00352 3/20 0.48
MAPK1 P28482 3/20 0.48
KDM4E B2RXH2 2/20 0.48
BLM P54132 1/20 0.48
TASP1 Q9H6P5 1/20 0.43
GAA P10253 2/20 0.42
HTT P42858 2/20 0.42
KCNJ6 P48051 2/20 0.42
KCNJ5 P48544 2/20 0.42
KCNJ3 P48549 2/20 0.42
POLB P06746 1/20 0.41
TP53 P04637 1/20 0.40
KMT2A Q03164 8/20 0.40
MEN1 O00255 6/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MMP13 P45452 1/20 0.40
LMNA P02545 2/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7920537 0.91 MAPT (0.46) MAPTALDH1A1MAPK1KDM4EBLM
SCHEMBL7922643 0.85 TASP1 (0.62) MAPTALDH1A1MAPK1KDM4ETASP1
SCHEMBL7922254 0.80 ALDH1A1 (0.44) MAPTALDH1A1MAPK1KDM4EBLM
SCHEMBL7922641 0.77 MAPT (0.61) MAPTALDH1A1MAPK1KDM4EBLM
SCHEMBL7922259 0.73 TASP1 (0.61) MAPTALDH1A1MAPK1KDM4ETASP1
SCHEMBL7922651 0.73 ALDH1A1 (0.59) MAPTALDH1A1MAPK1KDM4EBLM
SCHEMBL14096406 0.68 ALDH1A1 (0.54) MAPTALDH1A1MAPK1KDM4EBLM
SCHEMBL10069515 0.68 TASP1 (0.85) MAPTALDH1A1MAPK1KDM4EBLM
SCHEMBL14096409 0.67 ALDH1A1 (0.52) MAPTALDH1A1MAPK1KDM4EBLM
SCHEMBL19392442 0.61 KMT2A (0.54) MAPTALDH1A1MAPK1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100500-A1 THE USE OF CD4-BINDING SMALL MOLECULES TO INHIBIT HIV INFECTION THOMAS JEFFERSON UNIVERSITY (US) 2001-05-23 EP disclosed
WO-2000004903-A1 THE USE OF CD4-BINDING SMALL MOLECULES TO INHIBIT HIV INFECTION THOMAS JEFFERSON UNIVERSITY (US) 2000-02-03 WO disclosed