SCHEMBL7928260

SCHEMBL7928260

CCS(=O)(=O)c1ccc(-c2ccc3c(c2)C=C(C(=O)OC)CCS3(=O)=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.38
CA12 O43570 4/20 0.37
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
CA9 Q16790 4/20 0.37
KDM4E B2RXH2 1/20 0.34
CA14 Q9ULX7 3/20 0.34
RORC P51449 6/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
PTGS2 P35354 1/20 0.33
JAK2 O60674 1/20 0.32
PLAU P00749 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7972072 0.88 KIF11 (0.37) KIF11CA1CA2CA9KDM4E
SCHEMBL7934116 0.87 CTSL (0.39) CA12CA9ALDH1A1TSHRPOLB
SCHEMBL7975083 0.84 CA12 (0.39) CA12CA2CA9KDM4EALDH1A1
SCHEMBL7934057 0.84 SLC6A3 (0.40) CA12CA9KDM4EPTGS2ALDH1A1
SCHEMBL7922057 0.84 MAPT (0.42) KDM4EALDH1A1
SCHEMBL7971878 0.84 MCL1 (0.38) CA12CA9POLB
SCHEMBL7959206 0.84 POLB (0.34) CA12CA2CA9KDM4EPTGDR2
SCHEMBL7928263 0.84 F10 (0.34) PTGS2ALDH1A1POLB
SCHEMBL7969353 0.83 SLC6A3 (0.40) CA12CA2CA9KDM4EPLAU
SCHEMBL7934163 0.83 KDM4E (0.45) CA12CA1CA2CA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed