SCHEMBL7928263

SCHEMBL7928263

CCS(=O)(=O)c1ccccc1-c1ccc2c(c1)C=C(C(=O)OC)CCS2(=O)=O

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F10 P00742 2/20 0.34
ALOX5AP P20292 2/20 0.34
FEN1 P39748 2/20 0.34
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 3/20 0.33
PTGS2 P35354 1/20 0.33
SLC6A2 P23975 1/20 0.32
POLB P06746 1/20 0.32
SCN9A Q15858 2/20 0.31
ALDH1A1 P00352 1/20 0.31
ALOX12 P18054 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7972077 0.89 ALOX5AP (0.35) ALOX5APFEN1
SCHEMBL7928260 0.84 KIF11 (0.38) PTGS2POLBALDH1A1
SCHEMBL7959207 0.83 ALDH1A1 (0.34) ALOX5APFEN1SLC6A4SLC6A3SLC6A2
SCHEMBL7972215 0.82 PTGS2 (0.34) SLC6A4SLC6A3PTGS2SLC6A2POLB
SCHEMBL7972310 0.80 PTGS2 (0.37) SLC6A4SLC6A3PTGS2SLC6A2ALDH1A1
SCHEMBL7934116 0.79 CTSL (0.39) POLBALDH1A1
SCHEMBL7934057 0.77 SLC6A3 (0.40) SLC6A4SLC6A3PTGS2ALDH1A1
SCHEMBL7975083 0.77 CA12 (0.39) POLBALDH1A1HTT
SCHEMBL7959206 0.76 POLB (0.34) SLC6A4SLC6A3PTGS2SLC6A2POLB
SCHEMBL7971878 0.76 MCL1 (0.38) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed