SCHEMBL7950828

SCHEMBL7950828

NC(=O)CCCC(N)C(=O)c1nccs1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
PLA2G4A P47712 3/20 0.40
CES1 P23141 1/20 0.39
ALOX15 P16050 1/20 0.37
BLM P54132 1/20 0.37
PMP22 Q01453 1/20 0.37
KMT2A Q03164 1/20 0.37
F10 P00742 6/20 0.36
CTSK P43235 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
F2 P00734 2/20 0.34
F11 P03951 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8800894 0.94 ALDH1A1 (0.44) ALDH1A1PLA2G4ACES1ALOX15BLM
SCHEMBL7377556 0.86 ALDH1A1 (0.43) ALDH1A1PLA2G4ACES1F10CTSK
SCHEMBL7375810 0.85 GSR (0.43) ALDH1A1PLA2G4ACES1F10CTSK
SCHEMBL7378372 0.81 ALDH1A1 (0.42) ALDH1A1PLA2G4ACES1KMT2ACTSK
Hydrochloric Acid SCHEMBL28172161 0.81 PLA2G4A (0.40) ALDH1A1PLA2G4ACES1F10CTSK
SCHEMBL8801010 0.79 F10 (0.44) F10CTSKF2F11
SCHEMBL8802462 0.77 ALDH1A1 (0.44) ALDH1A1PLA2G4ACES1KMT2AF10
SCHEMBL27699627 0.76 ALDH1A1 (0.50) ALDH1A1PLA2G4ACES1
SCHEMBL7373337 0.76 ARG1 (0.64) ALDH1A1PLA2G4ACES1F10CTSK
SCHEMBL7373336 0.76 TBXAS1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6291678-B1 CAN BE INCORPORATED IN INHIBITORS OF SERINE PROTEASES WHICH ARE USED IN THERAPY OF ABNORMAL COAGULATION; THERAPY OR PROPHYLAXIS OF SEPTIC SHOCK, ATHEROSCLEROSIS, ALZHEIMER'S AND PARKINSON'S DISEASE WARNER-LAMBERT COMPANY 2001-09-18 US disclosed
EP-0906296-A1 PROCESS FOR THE PREPARATION OF CHIRAL KETO-HETEROCYCLES OF BASIC AMINO ACIDS WARNER-LAMBERT COMPANY LLC (US) 1999-04-07 EP disclosed
WO-1997048687-A1 PROCESS FOR THE PREPARATION OF CHIRAL KETO-HETEROCYCLES OF BASIC AMINO ACIDS WARNER-LAMBERT COMPANY (US) 1997-12-24 WO disclosed