SCHEMBL7952972

SCHEMBL7952972

CC(=O)c1c(C(F)(F)F)c(-c2cccnc2Cl)n2c1C(O)CCC2

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 10/20 0.34
NSD2 O96028 4/20 0.33
HCRTR2 O43614 2/20 0.33
CYP2C19 P33261 1/20 0.32
POLB P06746 1/20 0.32
ALDH1A1 P00352 1/20 0.32
DHODH Q02127 1/20 0.32
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7961238 0.90 ALDH1A1 (0.32) HCRTR1NSD2HCRTR2CYP2C19POLB
SCHEMBL7963301 0.90 HCRTR1 (0.34) HCRTR1NSD2CYP2C19POLBALDH1A1
SCHEMBL7965403 0.89 HCRTR1 (0.34) HCRTR1HCRTR2SCN9A
SCHEMBL7965010 0.87 HCRTR1 (0.33) HCRTR1HCRTR2CYP2C19POLBALDH1A1
SCHEMBL7965374 0.86 DHODH (0.36) HCRTR1HCRTR2CYP2C19ALDH1A1DHODH
SCHEMBL7952967 0.84 DPP4 (0.35) HCRTR1HCRTR2CYP2C19ALDH1A1DHODH
SCHEMBL7961656 0.83 FAAH (0.34) HCRTR1HCRTR2CYP2C19ALDH1A1DHODH
SCHEMBL7965321 0.83 KCNMA1 (0.34)
SCHEMBL7964875 0.80 CYP11B2 (0.37) HCRTR1HCRTR2ALDH1A1
SCHEMBL8327360 0.80 DHODH (0.35) HCRTR1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207675-B1 FOR PROPHYLAXIS AND THERAPY OF DISEASES IN WHICH ARE INVOLVED VIRUSES OF THE HERPES FAMILY AND/OR CYTOKINES IN PARTICULAR TUMOR NERCOSIS FACTOR-ALPHA RHONE-POULENC RORER S.A. (FR) 2001-03-27 US claimed
EP-0946555-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 1999-10-06 EP claimed
WO-1998025925-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM RHONE-POULENC RORER S.A. (FR) 1998-06-18 WO claimed
US-6207675-B1 FOR PROPHYLAXIS AND THERAPY OF DISEASES IN WHICH ARE INVOLVED VIRUSES OF THE HERPES FAMILY AND/OR CYTOKINES IN PARTICULAR TUMOR NERCOSIS FACTOR-ALPHA RHONE-POULENC RORER S.A. (FR) 2001-03-27 US disclosed