SCHEMBL7956997

SCHEMBL7956997

CN(C)CCOc1ccccc1Cc1nc(-c2ccccc2)no1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.58
DRD1 P21728 1/20 0.58
DRD4 P21917 1/20 0.58
DRD5 P21918 1/20 0.58
TSHR P16473 5/20 0.56
MAPK1 P28482 5/20 0.56
L3MBTL1 Q9Y468 5/20 0.56
TDP1 Q9NUW8 4/20 0.56
LMNA P02545 4/20 0.56
KDM4E B2RXH2 3/20 0.56
NPC1 O15118 6/20 0.52
RAB9A P51151 5/20 0.52
SMN1; SMN2 Q16637 5/20 0.52
MAPT P10636 3/20 0.52
HRH1 P35367 2/20 0.50
HTR7 P34969 1/20 0.50
HTR1A P08908 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963733 0.81 HTR7 (0.54) DRD2DRD1DRD4DRD5TSHR
Irampanel SCHEMBL678128 0.80 HTR7 (0.63) MAPK1L3MBTL1TDP1LMNAKDM4E
Irampanel SCHEMBL6879876 0.79 HTR7 (0.62) MAPK1L3MBTL1TDP1LMNAKDM4E
SCHEMBL7947527 0.78 RAB9A (0.57) TSHRMAPK1L3MBTL1TDP1LMNA
SCHEMBL7957012 0.77 NPC1 (0.49) TSHRMAPK1L3MBTL1TDP1LMNA
SCHEMBL7947228 0.76 HTR1A (0.73) TSHRMAPK1L3MBTL1TDP1NPC1
SCHEMBL5736045 0.75 HTR7 (0.63) TSHRL3MBTL1KDM4ENPC1RAB9A
Phenyltoloxamine SCHEMBL5145512 0.74 DRD1 (1.00) DRD2DRD1DRD4DRD5TSHR
Phenyltoloxamine SCHEMBL28854 0.74 DRD1 (1.00) DRD2DRD1DRD4DRD5TSHR
SCHEMBL7958685 0.73 NR1H4 (0.62) LMNAKDM4ENPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6277872-B1 ANTIISCHEMIC AGENTS; BRAIN DISORDERS BOEHRINGER INGELHEIM KG (DE) 2001-08-21 US disclosed