SCHEMBL7963780

SCHEMBL7963780

CC(C)c1ccc(OC(CCN2CCC(c3cnc4ccccc4n3)CC2)OC(=O)[C@H](O)c2ccccc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.37
AKT2 P31751 3/20 0.37
BCHE P06276 2/20 0.36
MAPT P10636 1/20 0.35
TP53 P04637 1/20 0.35
THRB P10828 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HRH1 P35367 3/20 0.34
ACACB O00763 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
LMNA P02545 1/20 0.34
MCHR1 Q99705 1/20 0.34
CCR5 P51681 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963779 0.83 MAPT (0.41) AKT1AKT2MAPTTP53MEN1
Mandelic Acid SCHEMBL7963777 0.77 MAPT (0.38) AKT1AKT2MAPTTP53MEN1
SCHEMBL23442934 0.64 AKT1 (0.44) AKT1AKT2MAPTTP53KMT2A
SCHEMBL25171674 0.64 HDAC4 (0.49) AKT1AKT2TP53LMNA
SCHEMBL7962234 0.62 HTR1A (0.36) AKT1AKT2
SCHEMBL7953579 0.61 CCR1 (0.41) MEN1KMT2ALMNA
SCHEMBL29891579 0.60 HPGDS (0.53) TP53THRBMEN1KMT2A
SCHEMBL3714809 0.60 HPGDS (0.53) TP53THRBMEN1KMT2A
SCHEMBL9074787 0.60 HTR1A (0.52) MCHR1
SCHEMBL24870232 0.58 HTR3A (0.49) BCHEMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed