SCHEMBL7966533

SCHEMBL7966533

O=C(OC1(c2cnc3ccccc3c2)CCN(CCCOc2ccccc2)CC1)C(=O)OC1(c2cnc3ccccc3c2)CCN(CCCOc2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
ALDH1A1 P00352 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.42
EGFR P00533 1/20 0.42
INSR P06213 1/20 0.42
IGF1R P08069 1/20 0.42
MET P08581 1/20 0.42
CDK2 P24941 1/20 0.42
KDR P35968 1/20 0.42
TEK Q02763 1/20 0.42
DRD3 P35462 4/20 0.41
DRD2 P14416 2/20 0.41
MMP1 P03956 2/20 0.41
MMP9 P14780 2/20 0.41
MMP13 P45452 2/20 0.41
ADAM17 P78536 1/20 0.41
HTR2A P28223 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7966503 0.85 MEN1 (0.46) KDM4EALDH1A1MEN1KMT2AIGF1R
Oxalic Acid SCHEMBL7966526 0.85 KDM4E (0.54) KDM4EALDH1A1SMN1; SMN2MEN1LMNA
SCHEMBL7962754 0.84 ALDH1A1 (0.56) KDM4EALDH1A1SMN1; SMN2MEN1LMNA
SCHEMBL7965014 0.84 OPRM1 (0.43) KDM4EALDH1A1SMN1; SMN2MEN1LMNA
SCHEMBL7966082 0.79 KDM4E (0.48) KDM4EALDH1A1SMN1; SMN2MEN1LMNA
SCHEMBL7964658 0.73 MEN1 (0.48) ALDH1A1MEN1LMNAKMT2AEGFR
Oxalic Acid SCHEMBL7966500 0.72 KMT2A (0.52) KDM4EALDH1A1MEN1LMNAKMT2A
Oxalic Acid SCHEMBL7965012 0.71 KDM4E (0.46) KDM4EALDH1A1SMN1; SMN2DRD3DRD2
SCHEMBL7966189 0.71 LTA4H (0.50) ALDH1A1MEN1LMNAKMT2AEGFR
Hydrochloric Acid SCHEMBL29427652 0.70 DRD3 (0.68) KDM4EALDH1A1SMN1; SMN2MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed
EP-0976747-A2 Use of 5HT-1F receptor antagonists for treating anxiety disorders ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed