SCHEMBL7972674

SCHEMBL7972674

COc1c2c(c(OC)c(OC)c1OC)CCC(CCOc1ccc3ccccc3n1)CC2

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 1/20 0.49
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
MCHR1 Q99705 2/20 0.38
FFAR1 O14842 1/20 0.34
HCRTR1 O43613 5/20 0.33
HCRTR2 O43614 5/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7961107 0.81 MEN1 (0.44) MEN1MAPTKMT2ADRD2DRD4
SCHEMBL7961186 0.80 HTR1A (0.43) DRD2DRD4BCHEACHE
SCHEMBL7972863 0.73 HRH3 (0.46) NPC1RAB9A
SCHEMBL7974660 0.71 CHRNB2 (0.46) DRD2
SCHEMBL27696506 0.70 MAPT (0.59) MEN1MAPTKMT2AKDM4ENPC1
SCHEMBL7977073 0.69 SIGMAR1 (0.44)
SCHEMBL30060467 0.68 MEN1 (0.61) MEN1MAPTKMT2AMCHR1KDM4E
SCHEMBL4269051 0.68 MEN1 (0.61) MEN1MAPTKMT2AMCHR1KDM4E
SCHEMBL7972868 0.68 HRH3 (0.41) ACHE
SCHEMBL4273391 0.67 MAPT (0.59) MEN1MAPTKMT2AMCHR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326369-B1 ALZHEIMER'S DISEASE TAKEDA CHEMICALS INDUSTRIES, LTD. (JP) 2001-12-04 US disclosed
EP-0968164-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2000-01-05 EP disclosed
WO-1998033758-A1 BICYCLIC QUINONE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-06 WO disclosed