SCHEMBL7977930

SCHEMBL7977930

O=C(O)c1nc(-c2ccccc2)[nH]c1-c1cccnc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 3/20 0.56
CYP1A2 P05177 1/20 0.56
MAPK1 P28482 1/20 0.56
CASP1 P29466 1/20 0.56
CYP2C19 P33261 1/20 0.56
RNASEH1 O60930 1/20 0.52
ERCC1 P07992 1/20 0.52
FEN1 P39748 1/20 0.52
ERCC4 Q92889 1/20 0.52
NPY5R Q15761 1/20 0.51
DHODH Q02127 3/20 0.50
KDM4E B2RXH2 2/20 0.50
LDHA P00338 1/20 0.50
EPHX2 P34913 1/20 0.50
HPGD P15428 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
STAT1 P42224 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29093221 0.86 PIN1 (0.69) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL7977705 0.85 DHODH (0.54) PIN1NPY5RDHODHKDM4ELDHA
SCHEMBL7992089 0.85 MAPK14 (0.62) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL7989683 0.82 ALDH1A1 (0.48) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL7988268 0.82 PIN1 (0.52) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL21652629 0.81 PIN1 (0.71) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL10649656 0.79 PIN1 (0.72) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL7978027 0.78 KDM4E (0.67) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL7372293 0.77 MKNK1 (0.58) CYP1A2CYP2C19NPY5RDHODHKDM4E
Hydrochloric Acid SCHEMBL7978210 0.77 RAB9A (0.53) CYP1A2MAPK1KDM4EHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288061-B1 INTERLEUKIN INHIBITORS; ASTHMA, BRONCHODILATOR AGENTS, ANTIALLERGENS WELFIDE CORPORATION (JP) 2001-09-11 US disclosed