SCHEMBL7979708

SCHEMBL7979708

CC1(C)C(=O)N(Cc2ccc(C#N)cc2)C(=O)c2cc(NS(=O)(=O)c3ccccc3)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.49
BRPF1 P55201 5/20 0.43
AR P10275 1/20 0.43
SMARCA2 P51531 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
DRD3 P35462 1/20 0.43
HTR6 P50406 1/20 0.43
IMPDH2 P12268 1/20 0.42
BRD4 O60885 4/20 0.41
CYP19A1 P11511 1/20 0.41
BRD1 O95696 3/20 0.41
BRD9 Q9H8M2 2/20 0.41
BRPF3 Q9ULD4 2/20 0.41
PGR P06401 1/20 0.41
MEN1 O00255 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7977859 0.83 F2 (0.49) TDP1
SCHEMBL7979527 0.77 TDP1 (0.51) TDP1HTR2CBRD4PGR
SCHEMBL7979619 0.74 TDP1 (0.48) TDP1CYP19A1PGR
SCHEMBL7479090 0.70 BRPF1 (0.52) BRPF1ARSMARCA2IMPDH2BRD4
SCHEMBL7572258 0.69 CYP19A1 (0.75) ARCYP19A1PGRMEN1KMT2A
SCHEMBL7428683 0.69 BRPF1 (0.52) BRPF1ARSMARCA2IMPDH2BRD4
SCHEMBL7981601 0.67 BRPF1 (0.51) BRPF1ARSMARCA2IMPDH2BRD4
SCHEMBL8029898 0.66 BRPF1 (0.61) BRPF1ARSMARCA2IMPDH2BRD4
SCHEMBL5784952 0.66 ADRA1D (0.64) BRD4KMT2A
SCHEMBL8028568 0.65 F2 (0.61) BRPF1ARSMARCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6200976-B1 FOR TREATING THROMBOSIS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-03-13 US disclosed