SCHEMBL7984973

SCHEMBL7984973

Oc1nc(-c2cccc(C(F)(F)F)c2)nc2ncn(Cc3ccccc3)c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 1/20 0.44
ADORA3 P0DMS8 2/20 0.43
GRIN2B Q13224 2/20 0.43
GRIN1 Q05586 1/20 0.43
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
ADORA2A P29274 1/20 0.41
ABCG2 Q9UNQ0 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
MMP13 P45452 1/20 0.39
PTPN1 P18031 1/20 0.38
PTPN6 P29350 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974072 0.94 ADORA3 (0.43) CXCR2ADORA3GRIN2BGRIN1ABCG2
SCHEMBL7988016 0.90 HDAC1 (0.44) ADORA3HDAC1HDAC6CTSSCTSK
SCHEMBL7987950 0.88 ADORA3 (0.49) CXCR2ADORA3ADORA2AABCG2ALDH1A1
SCHEMBL7987253 0.86 HPGDS (0.40) ADORA3HDAC1HDAC6ADORA2AABCG2
SCHEMBL7985336 0.85 PIK3CA (0.42) CXCR2ADORA3HDAC1HDAC6ADORA2A
SCHEMBL7975267 0.85 SMN1; SMN2 (0.46) ADORA3ADORA2AALDH1A1KMT2ASMN1; SMN2
SCHEMBL7974012 0.84 ALDH1A1 (0.41) CXCR2ADORA3HDAC1HDAC6ADORA2A
SCHEMBL7984659 0.84 ALDH1A1 (0.44) ADORA3ADORA2AALDH1A1KDM4EMEN1
Hydrochloric Acid SCHEMBL7987662 0.84 ALDH1A1 (0.43) ADORA3ADORA2AALDH1A1KDM4EMEN1
SCHEMBL7988594 0.84 TP53 (0.44) HDAC1HDAC6ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6310070-B1 FOR TREATING NEPHRITIS, IMPROVING PROTEINURIA DUE TO GLOMERULONEPHRITIS AND PREVENTING AGGRAVATION OF NEPHRITIS JAPAN ENERGY CORPORATION (JP) 2001-10-30 US disclosed
EP-0999211-A1 NOVEL PURINE DERIVATIVES AND MEDICINAL USE THEREOF JAPAN ENERGY CORPORATION (JP) 2000-05-10 EP disclosed