SCHEMBL7986050

SCHEMBL7986050

O=C(C1=Cc2cnc3cccc(n23)S1)N1CCC(CN2CCC(c3ccccc3)CC2)CC1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
CCR5 P51681 11/20 0.39
SCD5 Q86SK9 3/20 0.38
SCD O00767 1/20 0.38
CHRM4 P08173 2/20 0.37
OPRL1 P41146 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7986635 0.99 NPC1 (0.39) NPC1RAB9AKMT2ACCR5SCD5
SCHEMBL7982022 0.85 DRD2 (0.36) CCR5OPRL1KCNH2
Hydrochloric Acid SCHEMBL7983158 0.84 DRD2 (0.36) CCR5OPRL1KCNH2
SCHEMBL7983161 0.78 ALDH1A1 (0.43) KMT2AKCNH2
SCHEMBL7986651 0.78 USP5 (0.38)
SCHEMBL7982970 0.78 ADRA1D (0.45)
Hydrochloric Acid SCHEMBL7972919 0.77 ADRA1D (0.44)
Hydrochloric Acid SCHEMBL7971588 0.77 USP5 (0.38)
Hydrochloric Acid SCHEMBL7986162 0.77 ALDH1A1 (0.43) KMT2AKCNH2
SCHEMBL7984507 0.77 OGA (0.40) KMT2ACHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235731-B1 REDUCING BLOOD LIPIDS, SUGARS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0915888-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS Takeda Chemical Industries, Ltd. (JP) 1999-05-19 EP disclosed
WO-1997040051-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-30 WO disclosed