SCHEMBL7990500

SCHEMBL7990500

COc1ccc(-c2cncc(-c3cn(C(C)C4CCCNC4)c4ccc(C#N)cc34)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 6/20 0.41
CHEK1 O14757 2/20 0.37
PTPN11 Q06124 1/20 0.35
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNB3 Q05901 1/20 0.35
ALPL P05186 1/20 0.35
IKBKB O14920 1/20 0.34
CCNT1 O60563 1/20 0.34
CDK9 P50750 1/20 0.34
SCN9A Q15858 1/20 0.34
XDH P47989 1/20 0.34
TGFBR1 P36897 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987194 0.92 HTR6 (0.37) CHEK1CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL7990463 0.91 CHEK1 (0.39) KDM1ACHEK1SCN9A
SCHEMBL7994416 0.90 CCNT1 (0.37) KDM1ACHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL7505916 0.90 CCNT1 (0.38) KDM1ACCNT1CDK9
SCHEMBL7976151 0.88 CCNT1 (0.37) CHEK1CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL7986667 0.87 CDK7 (0.44) CHEK1CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL7990169 0.87 PDE4B (0.37) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL7990448 0.86 CYP11B1 (0.40) IKBKBCCNT1CDK9TGFBR1
SCHEMBL7993904 0.85 KDR (0.38) KDM1ACHEK1
SCHEMBL7975983 0.85 CCNT1 (0.36) KDM1ACCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed