SCHEMBL7991950

SCHEMBL7991950

CC1=NN(c2ccc3[nH]nnc3c2)C(=O)C(=O)C1=O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
PTGS2 P35354 1/20 0.32
KAT8 Q9H7Z6 3/20 0.31
AMY1A P0DUB6 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7985940 0.76 IDO1 (0.44) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL7985908 0.70 MAPT (0.35) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL7989137 0.69 POLB (0.41) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL23348987 0.69 POLB (0.44) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL9717736 0.68 L3MBTL1 (0.40) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL23348985 0.68 CA12 (0.39) KDM4EGAA
SCHEMBL7989367 0.68 PTGS2 (0.43) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL6736416 0.67 KMT2A (0.49) ALDH1A1KDM4EMEN1GAAMAPT
SCHEMBL29367601 0.65 CYP1A2 (0.39) ALDH1A1GAAKMT2A
SCHEMBL103309 0.65 CYP1A2 (0.39) ALDH1A1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271373-B1 PYRIDINE DERIVATIVE FORMED BY REACTING A PYRAZINE DERIVATIVE WITH FECL3 AND ACETIC ACID VIROPHARMA INCORPORATED 2001-08-07 US disclosed
US-6180628-B1 PYRIDAZINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH DERIVATIVES AND THEIR USE IN TREATING INFLUENZA INFECTION AND OTHER VIRAL DISEASES VIROPHARMA INCORPORATED 2001-01-30 US disclosed
EP-0920419-A4 COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATING INFLUENZA VIROPHARMA INC (US) 1999-10-06 EP disclosed
US-5935957-A PYRIDAZINE DERIVATIVES VIROPHARMA INCORPORATED (US) 1999-08-10 US disclosed
EP-0920419-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATING INFLUENZA Viropharma Incorporated (US) 1999-06-09 EP disclosed
US-5821243-A 3,4,5-TRIOXO-2H,3H,4H,5H-PYRIDAZINES; TRANSCRIPTASE INHIBITORS; NONTOXIC VIROPHARMA INCORPORATED (US) 1998-10-13 US disclosed
WO-1998003487-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATING INFLUENZA VIROPHARMA INCORPORATED (US) 1998-01-29 WO disclosed