SCHEMBL7993465

SCHEMBL7993465

CC(C)(C)OC(=O)N1CC[C@@H](NS(=O)(=O)c2cc(N)ccc2Cl)C1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.51
STS P08842 4/20 0.49
SFRP1 Q8N474 3/20 0.47
CCR8 P51685 1/20 0.46
USP30 Q70CQ3 2/20 0.45
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NR1H2 P55055 1/20 0.44
EPHX2 P34913 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8022249 0.91 STS (0.53) BRD4STSSFRP1CCR8USP30
SCHEMBL8023062 0.87 SFRP1 (0.51) BRD4STSSFRP1CCR8
SCHEMBL7982132 0.87 STS (0.57) BRD4STSSFRP1CCR8USP30
SCHEMBL8004225 0.85 L3MBTL1 (0.50) BRD4STSSFRP1CCR8ALDH1A1
SCHEMBL3813973 0.85 ACLY (0.45) SFRP1ALDH1A1L3MBTL1
SCHEMBL4734403 0.80 STS (0.54) BRD4STSSFRP1CCR8
SCHEMBL4618399 0.78 SFRP1 (0.70) SFRP1CCR8
SCHEMBL8015057 0.78 USP30 (0.57) BRD4STSSFRP1CCR8USP30
SCHEMBL1320324 0.78 STS (0.55) BRD4STSSFRP1CCR8NPC1
SCHEMBL6194827 0.78 STS (0.55) BRD4STSSFRP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090264499-A1 Cathepsin C Inhibitors GLAXO GROUP LIMITED (GB) 2009-10-22 US disclosed
WO-2009129371-A1 CATHEPSIN C INHIBITORS GLAXO GROUP LIMITED (GB) 2009-10-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090264499-A1 Cathepsin C Inhibitors CTSB, CTSF, CTSG BRD4 1848/4885STS 3498/4885SFRP1 3908/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.