SCHEMBL7997927

SCHEMBL7997927

Nc1ccc(S(=O)(=O)Nc2cccc(OBOc3cccc(NS(=O)(=O)c4ccc(N)cc4)c3)c2)cc1

nearest known ligand 0.72

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.66
CA1 P00915 2/20 0.61
CA2 P00918 2/20 0.61
KMT2A Q03164 1/20 0.58
CYP19A1 P11511 2/20 0.52
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
KEAP1 Q14145 1/20 0.50
PKM P14618 1/20 0.50
HPGD P15428 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HTT P42858 1/20 0.49
CA9 Q16790 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8010004 0.87 POLB (0.64) HTR6CA1CA2KMT2ACYP19A1
SCHEMBL2242644 0.84 HTR6 (0.72) HTR6CA1CA2KMT2ACYP19A1
SCHEMBL8013124 0.82 CA2 (0.61) CA1CA2KMT2ACYP19A1ALDH1A1
SCHEMBL8018878 0.82 POLB (0.59) CA1CA2KMT2ACYP19A1ALDH1A1
SCHEMBL11438430 0.81 HTR6 (0.62) HTR6CA1CA2KMT2ACYP19A1
SCHEMBL8007630 0.80 POLB (0.56) CA1CA2KMT2AALDH1A1CA9
SCHEMBL28271812 0.80 HTR6 (1.00) HTR6CA1CA2KMT2ACYP19A1
SCHEMBL8013318 0.79 POLB (0.55) CA1CA2KMT2AALDH1A1CA9
SCHEMBL8010014 0.78 PGR (0.65) HTR6CA1CA2KMT2AALDH1A1
SCHEMBL24125035 0.76 HTR6 (0.73) HTR6CA1CA2KMT2ACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000035904-A1 INHIBITORS OF β-LACTAMASES AND USES THEREFOR NORTHWESTERN UNIVERSITY (US) 2000-06-22 WO disclosed