SCHEMBL8024571

SCHEMBL8024571

O=C(O)CN(C(=O)C(CS)CCc1ccccc1)c1ccc(OCc2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.46
FFAR4 Q5NUL3 2/20 0.46
MMP12 P39900 1/20 0.44
SERPINE1 P05121 1/20 0.43
MRGPRX4 Q96LA9 2/20 0.43
MAOB P27338 1/20 0.41
KEAP1 Q14145 1/20 0.40
MLYCD O95822 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
ALOX5 P09917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8024336 0.92 FFAR1 (0.50) FFAR1FFAR4MMP12MAOBKEAP1
SCHEMBL8020340 0.91 MMP12 (0.48) FFAR1FFAR4MMP12MAOBKEAP1
SCHEMBL8010235 0.89 MMP12 (0.47) FFAR1FFAR4MMP12MAOBKEAP1
SCHEMBL8026747 0.88 ALOX5 (0.52) FFAR1FFAR4MMP12MAOBALOX5
SCHEMBL8010404 0.88 FFAR1 (0.49) FFAR1FFAR4MMP12MAOBKEAP1
SCHEMBL8026644 0.88 NOX1 (0.52) FFAR1FFAR4MMP12MAOBKEAP1
SCHEMBL8021316 0.86 NPC1 (0.49) FFAR1FFAR4MMP12MAOBKEAP1
SCHEMBL8021221 0.84 MEN1 (0.48) FFAR1FFAR4MMP12MAOBKEAP1
SCHEMBL8024296 0.84 NOX1 (0.48) MMP12MAOB
SCHEMBL8024699 0.84 FFAR1 (0.43) FFAR1FFAR4MMP12MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US claimed
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed