SCHEMBL8026644

SCHEMBL8026644

CN(C)c1ccc(COc2ccc(N(CC(=O)O)C(=O)C(CS)CCc3ccccc3)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 1/20 0.52
MAOB P27338 4/20 0.48
MMP12 P39900 1/20 0.46
FFAR1 O14842 1/20 0.46
FFAR4 Q5NUL3 1/20 0.46
LTB4R Q15722 1/20 0.44
LTB4R2 Q9NPC1 1/20 0.44
ALOX5 P09917 1/20 0.43
KEAP1 Q14145 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8024336 0.95 FFAR1 (0.50) MAOBMMP12FFAR1FFAR4ALOX5
SCHEMBL8020340 0.94 MMP12 (0.48) NOX1MAOBMMP12FFAR1FFAR4
SCHEMBL8023120 0.92 FFAR1 (0.46) NOX1FFAR1LTB4RLTB4R2KEAP1
SCHEMBL8010404 0.92 FFAR1 (0.49) MAOBMMP12FFAR1FFAR4KEAP1
SCHEMBL8010235 0.92 MMP12 (0.47) MAOBMMP12FFAR1FFAR4ALOX5
SCHEMBL8026747 0.90 ALOX5 (0.52) MAOBMMP12FFAR1FFAR4ALOX5
SCHEMBL8024296 0.89 NOX1 (0.48) NOX1MAOBMMP12
SCHEMBL8021316 0.88 NPC1 (0.49) NOX1MAOBMMP12FFAR1FFAR4
SCHEMBL8024571 0.88 FFAR1 (0.46) MAOBMMP12FFAR1FFAR4ALOX5
SCHEMBL8021221 0.87 MEN1 (0.48) MAOBMMP12FFAR1FFAR4KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US claimed
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed