SCHEMBL8024296

SCHEMBL8024296

CC(=O)Nc1ccc(COc2ccc(N(CC(=O)O)C(=O)C(CS)CCc3ccccc3)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 2/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
POLB P06746 2/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
LTA4H P09960 5/20 0.44
CASP3 P42574 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
GPR55 Q9Y2T6 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8024336 0.92 FFAR1 (0.50) MAOBMMP12
SCHEMBL8020340 0.91 MMP12 (0.48) NOX1MAOBMMP12
SCHEMBL8026644 0.89 NOX1 (0.52) NOX1MAOBMMP12
SCHEMBL8010404 0.89 FFAR1 (0.49) MEN1KMT2AMAOBMMP12
SCHEMBL8010235 0.89 MMP12 (0.47) LMNAMAOBMMP12
SCHEMBL8026747 0.87 ALOX5 (0.52) SMN1; SMN2NPC1RAB9APOLBMAOB
SCHEMBL8021316 0.85 NPC1 (0.49) NOX1SMN1; SMN2NPC1HTTMAOB
SCHEMBL8024571 0.84 FFAR1 (0.46) MAOBMMP12
SCHEMBL8021221 0.84 MEN1 (0.48) MEN1KMT2ASMN1; SMN2ALDH1A1LMNA
SCHEMBL8010401 0.84 ALDH1A1 (0.45) NOX1MEN1KMT2ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US claimed
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed