SCHEMBL8019501

SCHEMBL8019501

C=C(c1ccc(NC(=O)c2ccc(S(C)(=O)=O)cc2)cc1S(=O)(=O)O)c1ccc(NC(=O)c2ccc(S(C)(=O)=O)cc2)cc1S(=O)(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.56
ADORA2A P29274 1/20 0.56
ADORA2B P29275 1/20 0.56
ADORA1 P30542 1/20 0.56
AVPR2 P30518 1/20 0.47
GPR27 Q9NS67 1/20 0.47
RORC P51449 1/20 0.46
LRRK2 Q5S007 1/20 0.45
RAD51 Q06609 1/20 0.44
LMNA P02545 1/20 0.44
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
ROCK2 O75116 1/20 0.43
SIRT2 Q8IXJ6 1/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 1/20 0.43
ENPP2 Q13822 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8021833 0.88 ADORA3 (0.43) ADORA3ADORA2AADORA2BADORA1RORC
SCHEMBL8008341 0.84 MEN1 (0.45) ADORA3ADORA2AADORA2BADORA1RAD51
SCHEMBL8008740 0.83 ENPP2 (0.39) ADORA3ADORA2AADORA2BADORA1RAD51
SCHEMBL8023363 0.82 ADORA3 (0.56) ADORA3ADORA2AADORA2BADORA1RORC
SCHEMBL8019113 0.82 RAD51 (0.40) ADORA3ADORA2AADORA2BADORA1RORC
SCHEMBL8021340 0.82 VCAM1 (0.55) LMNAMEN1KMT2AALDH1A1NPC1
SCHEMBL7665070 0.81 RAD51 (0.59) ADORA3ADORA2AADORA2BADORA1RORC
SCHEMBL7678186 0.81 ADORA3 (0.57) ADORA3ADORA2AADORA2BADORA1RORC
SCHEMBL7665009 0.81 RAD51 (0.59) ADORA3ADORA2AADORA2BADORA1RORC
SCHEMBL9359160 0.78 ENPP2 (0.57) CA1CA2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000058277-A1 ARYL SULFONIC ACIDS AND DERIVATIVES AS FSH ANTAGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 2000-10-05 WO claimed
WO-2000058277-A1 ARYL SULFONIC ACIDS AND DERIVATIVES AS FSH ANTAGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 2000-10-05 WO disclosed