SCHEMBL8024858

SCHEMBL8024858

COCOc1cccnc1C(=O)c1ccc(F)c(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
HPGD P15428 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B14 Q9BPX1 1/20 0.36
APAF1 O14727 1/20 0.36
NSD2 O96028 1/20 0.36
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PDE10A Q9Y233 2/20 0.36
EGFR P00533 1/20 0.36
NPC1 O15118 1/20 0.34
MAPK1 P28482 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ADORA2A P29274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709579 0.84 KDM4E (0.38) ALDH1A1CYP2D6CYP2C19APAF1NSD2
SCHEMBL8020333 0.83 XDH (0.45) ALDH1A1HPGDCYP1A2CYP2D6CYP2C19
SCHEMBL8020675 0.82 TDP1 (0.42) ALDH1A1HPGDCYP1A2CYP2D6CYP2C19
SCHEMBL8023521 0.79 HSD17B14 (0.50) HSD17B14
SCHEMBL8709890 0.78 RAB9A (0.37) ALDH1A1HPGDNPC1ADORA2AKDM4E
SCHEMBL8714963 0.77 PPIA (0.43) ALDH1A1HPGDL3MBTL1NPC1MAPK1
SCHEMBL8709054 0.75 CYP3A4 (0.47) ALDH1A1CYP2D6CYP2C19KDM4EMAPT
SCHEMBL8715277 0.74 CLCN2 (0.38) ALDH1A1APAF1NSD2CASP3SENP8
SCHEMBL8712836 0.74 MAPK8 (0.37) ALDH1A1HPGDL3MBTL1NPC1MEN1
SCHEMBL8713191 0.74 MAPK8 (0.39) ALDH1A1HPGDL3MBTL1NPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802187-B1 Hydroxypyridine derivatives, their production and their pharmaceutical use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-02-16 EP disclosed
US-5891895-A POTASSIUM CHANNEL MODULATORS; ANGINA PECTORIS; HYPERTENSIVEAGENTS; CARDIOVASCULAR, RESPIRATORY SYSTEM, BRAIN, GASTROINTESTINAL AND UROGENITAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US disclosed
EP-0802187-A1 Hydroxypyridine derivatives, their production and their pharmaceutical use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-22 EP disclosed